that is why i am curious that if IM/SC injection works to rapidly deliver diazepam, i dont see why IN avizafone should be any different. maybe sublingual, too
I read a medical journal that studies the IN administration of super saturated Avizafone (human enzym peptide to convert pro-drug into API Diazepam) it worked very well and is a promising alternative to future drugs to combat cluster seizures and other medical conditions requiring rapid sedation/muscle relaxation/anticonvulsant etc. Just google it in and you’ll find the IN study. This is the main study I read prior….
This is the real data from the study published in the medical journal…
National Library of Medicine - British Journal of Pharmacology
Bioavailability of Diazepam after intramuscular injection of its water-soluble prodrug Avizafone or Diazepam itself
The aim of this study was to assess the relative bioavailability of diazepam after administration of diazepam itself or as a water-soluble prodrug, avizafone, in humans.
C-Max (ng’mL-1)
Avizafone 223 (reaches MUCH higher levels in CNS - basically double)
Diazepam 118
T-Max (h)
Avizafone 0.76 (MUCH faster to achieve full concentration)
Diazepam 1.5
AUC 0-t (h
Avizafone 5584
Diazepam 5224
Probably the best prodrug ever synthasized …..Avizafone (Pro-Diazepam) rapid acting, water soluble, prodrug IM injection entering bloodstream were Typsin cleaves prodrug molecule into Lysin and the API, being Diazepam (Valium)
Avizafone (Pro-Diazepam) 4,000mg procured over several years …..light yellow, sticky powder sensitive to light, heat and moisture. MUST keep in fridge crisper drawer.
Oral administration is bullshit……IM injection is the only way. Sorry. Just ask the pharmacist for a 1ml syringe for IM administration, a 1inch needle most likely, into the shoulder muscle. Use once, they’re so cheap and so sharpe you won’t feel it
Add hot water into small glass vial with Avizafone 40-80mg, shake and swirl around to dissolve properly into a light yellow solution, no filter required, just draw up, prep it, no air etc, shoulder muscle, pop, break the skin and slowly glide that razor sharpe needle deep into the shoulder muscle…..press the plunger down.
In 10-15min you’ll feel the onset creeping in, you’ll even taste it in your mouth (strange I Know)
Before you’ll know it, you’ll melt into the couch with robust anxiolytic & muscle relaxant properties
Diazepam (Valium)
Methylphenidate (Ritalin)
Phenmetrazine (Preludin)
Amph salts (Biphetamine)
d-Amphetamine (Dexedrine)
d-Methamphetamine (Desoxyn/Methedrine)
Dexamyl & Desbutal
Methadone/Oxycodone/Diacetylmorphine/Hydromorphine
Didrex (Pro-Drug) metabolizes into d-Methamphetamine and then finally into d-Amphetamine
Vyvanse (Lisdexamfetamine) pro-drug metabolizing into active d-Amphetamine
Avizafone (Pro-Diazepam) prodrug metabolizing into Diazepam (Valium)
Diclazepam (pro-drug) metabolizes into 3 Pharma Benzo’s > Diclazepam >> Lorazepam (Ativan)
I just want a professional state of the art pharmaceutical laboratory synthesizing every CII substance known to man….relics from the 1950’s. There are secure drug houses with 100kg (220lbs) blue plastic drums of various CII chemicals, example Methadone Hydrochloride, Pregabalin HCL, etc even Cocaine Hydrochloride in 25gram glass jars labelled “light fluffy crystals” Warning: May be habit forming lol…..Fck me silly
Diacetylmorphine (Heroin) ..there are several closely related drugs Sooooo much better, faster acting, more potent, and longer lasting …..there is such an impressive list of analogs and similar opioid narcotics
Methedrine (d-N-Methyl Amphetamine Hydrochloride) 20 & 30mg glass vials for IV/IM/SC injection
Desoxyn 5mg tablets currently marketed
To be the head president of restricted CII controlled substances in the 1950’s with production runs producing millions of pressed branded tablets and raw API compounding powder ….fuuuuuuu ck
