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Drug designs. (MedicinalUser SAR thread)

On imgur you can change viewer links to BBcode full, then you can add the pictures on this site using the image button.

That way people don't have to click on every link.

Or like this without the spaces:

[ img]https://i.ibb.co/grS2D5r/start-44.png[ /img]

start-44.png
 
I know of a good piperazine that is active called 2-benzhydrylpiperazine.

Jongh David Karel De, Akkerman Antonie Marie, Kofman Hendrik,& Vries George De, U.S. patent 2,997,473 (1961 to Nederlandsche Combinatie voor Chemische Industrie NV).
Karel De Jongh David, et al. GB 893391 (1962 to Nederlandsche Combinatie voor Chemische Industrie NV).

I'd recommend this one to you. It's a central stimulant.
 
MedicinalUser247 said:
I call this one Magic Dust. https://ibb.co/P1v5qtp
Click to expand...
Have you seen

GK-189
1-[1-(2-Naphthalenyl)cyclohexyl]-Piperidine
[81490-58-6]

Apparently similar to BTCP, affecting catecholaminergic neurotransmission circuitry. 36nM for DA & 8nM for NE.

[1] Jean-Marc Kamenka, et al. US5248686 (1993 to Centre National de la Recherche Scientifique CNRS).
[2] Fotadar, Upinder Indian Journal of Chemistry, Section B: Organic Chemistry Including Medicinal Chemistry, 1981 , vol. 20, # 11 p. 1006 – 1007.
[3] Ilagouma, AT; Maurice, T; Duterte-Boucher, D; Coderc, E; Vignon, J; Costentin, J; Kamenka, JM (1993). "Arylcyclohexylamines derived from BTCP are potent indirect catecholamine agonists". European Journal of Medicinal Chemistry. 28 (5): 377–385. doi:10.1016/0223-5234(93)90124-W.
 
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