Coaxil and the Crocodile: Post-Soviet Heroin Substitutes

Kenaz

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The first post to my new blog, Opiated Shamanism. I've removed the links: you can find them on the blog, although I don't recommend clicking on some of the graphic images at work or on a full stomach.

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(Thanks to Bugsy of Opiophile and Dankycodone of Bluelight for pointing me toward some primary sources!)


The former Soviet Republics have seen better days - and even those weren't particularly good. Between the Berlin Wall's collapse and 2001, the average ex-comrade's buying power decreased nearly 25% in Russia, approximately 60% in Georgia, and over 80% in Tajikistan. The social services provided by the Party (such as they were) got swept aside in the new rush to economic freedom: the entrenched culture of corruption and oppression remained firmly in place. A few plutocrats became richer while most of the populace got a whole lot poorer.

Seeking solace or anesthesia, many turned to drugs. Today much of the region is awash in cheap Afghan heroin, imported through Uzbekistan, Kyrgyzstan, Tajikistan and Kazakhstan. But many users who lack the means to support a heroin habit - or who would rather avoid harsh penalties and legal harassment - have discovered new ways to abuse drugs which are readily available at their local pharmacies.

Antidepressants like Prozac and Paxil act as SSRIs, selective serotonin reuptake inhibitors. They interfere with the brain's uptake of serotonin, thereby leaving more available at the synapses to stimulate the receptors. Tianeptine, the active ingredient in the Russian antidepressent Coaxil, has the opposite effect: it encourages uptake and decreases extracellular serotonin levels. Nobody is sure why this also alleviates depression, or indeed, how tianeptine works within the human brain. But some experimentally-minded addicts have discovered that it also has a pronounced effect on the opiate receptors. Users compare intravenous Coaxil to a slightly speedier heroin shot, with a euphoric if somewhat short-lasting rush.

Alas, these effects only appear at a comparatively high dosage. A Coaxil tablet contains 12.5 milligrams of tianeptine: to get high, users shoot dozens of pills. The resulting solution is filled with insoluble particulates. Most Coaxil abusers use large needles to avoid clogging: this causes damage upon the first venipuncture and results in greater quantities of thrombosis-causing gunk pouring into the circulatory system. Abscesses and gangrene are common: amputations are frequently required.

Other addicts start with codeine tablets, which are widely available in most pharmacies. After crushing the pills, they engage in a multi-step chemical process akin to the making of "bathtub meth." Iodine and red phosphorous from match heads is added to solvents in an effort to transform the codeine into desomorphine, a powerful analog 10 times stronger than morphine.

The end result of this process contains some desomorphine: it also contains codeine and large amounts of iodine, phosphorous, acids and other toxic chemicals. Russians call it "the Crocodile" because users soon develop open sores, peeling and ulcers on their roughened skin. The liquid is highly corrosive and acidic, causing enormous damage to the circulatory system. Excessive iodine poisons the kidneys, thyroid and liver: excessive phosphorous can cause brain damage and necrosis of the jawbone, known among 19th century matchmakers as "phossy jaw." Intravenous codeine can cause pulmonary edema and histaminic shock. And because desomorphine is a relatively fast-acting opiate, users tend to inject repeatedly, thereby magnifying the consequences of each dose.
 
Other addicts start with codeine tablets, which are widely available in most pharmacies. After crushing the pills, they engage in a multi-step chemical process akin to the making of "bathtub meth." Iodine and red phosphorous from match heads is added to solvents in an effort to transform the codeine into desomorphine, a powerful analog 10 times stronger than morphine.

meth? that doesnt make sense...
 
How doesn't it make sense? They are comparing it to making meth in terms of household items and setup.. akin = similar
 
Homebake is more of making a heroin-ish substance out of poppy straw.. but I get what you're saying.

Crocodile-cooking is like Oceania's "homebake" in that it starts with codeine tablets. But homebake chemists try to transform methylmorphine (aka codeine) into plain old morphine, then add some AA to make it diacetylmorphine. The Russian DIY chemists are trying to make desomorphine. Their process uses iodine and red phosphorus, ingredients which, to the best of my knowledge, don't appear in the homebake recipe.

Ever get iodine on a cut or a scrape? Imagine how it feels in a vein. And I can't imagine phosphorus, IV codeine, or any of the other solvents used would be any more pleasant.
 
Are you certain that they're using HI/RP?

I'd imagine it could address that hydroxyl, but i'm less confident in it's ability to saturate the double bond....

And then there's the pesky problem of demethylating it.

I suspect different chemistry than that used to make meth is being used.

However, it seems like this is a relatively easy synthetic process, even if it's not as simple as they're letting on - one wonders why desmorphine isn't all over the illicit market. Hell, why does anyone make heroin out of opium, when they could be making desmorphine, cleaning up better than the russians do, and cutting it? For that matter, why not acetylate the desmorphine, yielding, if you will, "desheroin"? Would probably be even more recreational than desmorphine, and just as potent.


In any case, i've gotta say, it's scary to read about just how far opiate addicts will go for their fix when under desperate living conditions.
 
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As usual, a very interesting read. Nice work Kenaz, thanks.

Thanks. I'm hoping to keep the blog updated regularly between now and the release of my book. Between talking about junkies famous and otherwise and opiates in different cultures, I should be able to stay busy for a while.

Russia is a great example of just how effective a punitive/moralistic approach to drug addiction really is. Their cops have powers our DEA agents could only dream about, and they can't stop people from shooting up antidepressants and iodine solutions.
 
^great peice, man! I added your blog to my news readers so I hope you do keep updating it.

I wasn't sure if this would be best suited in OD or elsewhere so I conferred with other staff and its been decided that It's better suited for the DitM forum so we'll send it over there.


--->DitM
 
A bit of time ago I saw a bunch of videos about the sad state that heavy desomorphine users are in. I had no idea what the videos were saying since they weren't in english, and I'm not sure if the damage was caused by bad iv technique or the drug itself. Probably a mixture of both. Still, they were truly terrifying images...
 
A bit of time ago I saw a bunch of videos about the sad state that heavy desomorphine users are in. I had no idea what the videos were saying since they weren't in english, and I'm not sure if the damage was caused by bad iv technique or the drug itself. Probably a mixture of both. Still, they were truly terrifying images...

if you remember a link and theyre in russian id be glad to translate. but heroin is a huge problem in russia and belarus, i was in belarus a couple summers ago. talked with local kids and such and after alcohol i assume heroin would be 2nd or 3rd in popularity. id also hear about crazy ass ways these kids would get high, innovation at its saddest and finest points.
 
Red Phosphorus is not in match tips, it is in the match stiker pads on the box or matchbook..at least i nthe US it is..sulphur and othe rshit is actually in the matchtip itself and the Red P is in the stike pad ,a common misconception held by many people is that matchtips are a source for Red P ,but it is the stiking pad that is scrapped off a matchbook or box which contains the Red P,as any meth cook that used match books to obtain their dirty "Red P" ,the stike pad also has sandy shit to make it gritty,which often is not filtered in some small Red P meth labs..other than that good article..
 
if you remember a link and theyre in russian id be glad to translate. but heroin is a huge problem in russia and belarus, i was in belarus a couple summers ago. talked with local kids and such and after alcohol i assume heroin would be 2nd or 3rd in popularity. id also hear about crazy ass ways these kids would get high, innovation at its saddest and finest points.

http://www.youtube.com/watch?v=Cr_rdhiUznA

Here's one I just found, there's a bunch more out there that are more graphic. Don't worry about spending time translating though, the images speak loud enough.
 
^great peice, man! I added your blog to my news readers so I hope you do keep updating it.

I wasn't sure if this would be best suited in OD or elsewhere so I conferred with other staff and its been decided that It's better suited for the DitM forum so we'll send it over there.


--->DitM

Glad you enjoyed it. Does anyone object if I include other posts here? I'm working on a post on TimeRX, Oxy OP and other "anti-abuse" systems which will probably be a bit basic for Bluelight, but my next post describing the heroin scene in Yunnan, China (conveniently located between Burma and Afghanistan) may prove interesting to BL readers.

I don't want to become Spammy McSpammer flooding the boards with links to my blog and promos for my book. If you would rather I keep posts to a minimum let me know.
 
Red Phosphorus is not in match tips, it is in the match stiker pads on the box or matchbook..at least i nthe US it is..sulphur and othe rshit is actually in the matchtip itself and the Red P is in the stike pad ,a common misconception held by many people is that matchtips are a source for Red P ,but it is the stiking pad that is scrapped off a matchbook or box which contains the Red P,as any meth cook that used match books to obtain their dirty "Red P" ,the stike pad also has sandy shit to make it gritty,which often is not filtered in some small Red P meth labs..other than that good article..

Thanks. That's good to know: I've made the appropriate edit here and on my blog!
 
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