endotropic
Bluelight Crew
- Joined
- Feb 14, 2012
- Messages
- 1,140
Fentanyl
- μ - Mu = Affinity: .7nM Activity: ?
- κ - Kappa = Affinity: 84.8nM Activity: ?
- δ - Delta = Affinity: 152.7nM Activity: ?
I'll edit my post with the efficacy information later
Edit: what outcome are we using to determine activity? analgesic effect in people? GTPgammaS stimulation? AC inhibition? whatever we feel like?
- μ - Mu = Affinity: .7nM Activity: ?
- κ - Kappa = Affinity: 84.8nM Activity: ?
- δ - Delta = Affinity: 152.7nM Activity: ?
I'll edit my post with the efficacy information later
Edit: what outcome are we using to determine activity? analgesic effect in people? GTPgammaS stimulation? AC inhibition? whatever we feel like?
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