its called tofisopam
wikipedia:
Tofisopam (marketed under brand names Emandaxin and Grandaxin) is a drug which is a benzodiazepine derivative. Like other benzodiazepines, it possesses anxiolytic properties but not anticonvulsant, sedative,[1] skeletal muscle relaxant, motor skill-impairing or amnestic[2] properties. While it may not be an anticonvulsant in and of itself, it has been shown to enhance the anticonvulsant action of classical 1,4-benzodiazepines such as diazepam (but not sodium valproate, carbamazepine, phenobarbital, or phenytoin).[3]
Tofisopam is not approved for sale in the United States or Canada. However, Vela Pharmaceuticals of New Jersey is developing the D- enantiomer (dextofisopam) as a treatment for irritable bowel syndrome.[4]
and 1 user experience i found on the net
I tried it while living in Egypt :
It comes in 50mg and the usual effect lasts 5 hours.It is usually taken in 100mg 3 times daily,and is not recomended to be taken befoe bedtime because it is the only "STIMULANT BENZODIAZEPINE" on the planet.
My experience is that it gives you a relaxed feeling combined with excellent concentration,motivation and sociability,without any muscle relaxant or any sedative,amnestic proporties + NO withdrawal effects at all
Its structure is fundementaly different from any other BZ (2,3 benzo) and,from my own experience I believe that it must be affecting dopamine in a way
The great thing about it is that you can take as needed for focus + anxiety or chronically without worrying about withdrawal.....
I know I might sound talking about a fantasy drug ,but the truth is that I only stopped it because I left Egypt and could not find it in the other countries I lived in......
Acta Pharm Hung. 1993 Mar;63(2):91-8.
Excerpts from the clinical-pharmacologic and clinical studies of Grandaxin
Szego J, Somogyi M, Papp E.
EGIS Gyogyszergyar Rt., Budapest.
The authors give a selection from the clinical-pharmacological and clinical studies of Grandaxin (tofizopam), an original Hungarian compound registered in 1976. Tofizopam, a 2,3-benzodiazepine derivative, differs from "classical" 1,4-benzodiazepines not only in chemical structure, but also in pharmacological and clinical-pharmacological properties. It is an anxiolytic without sedative-hypnotic, muscle relaxant and anticonvulsive effects. Tofizopam does not impair psychomotor and intellectual performance, like other benzodiazepines do, in the contrary, it has a mild stimulatory activity. It is potent in alleviating vegetative symptoms accompanying anxiety disorders. Tofizopam has a very low toxicity, mild side effects. The administration of tofizopam does not lead to physical or psychic dependence.
wikipedia:
Tofisopam (marketed under brand names Emandaxin and Grandaxin) is a drug which is a benzodiazepine derivative. Like other benzodiazepines, it possesses anxiolytic properties but not anticonvulsant, sedative,[1] skeletal muscle relaxant, motor skill-impairing or amnestic[2] properties. While it may not be an anticonvulsant in and of itself, it has been shown to enhance the anticonvulsant action of classical 1,4-benzodiazepines such as diazepam (but not sodium valproate, carbamazepine, phenobarbital, or phenytoin).[3]
Tofisopam is not approved for sale in the United States or Canada. However, Vela Pharmaceuticals of New Jersey is developing the D- enantiomer (dextofisopam) as a treatment for irritable bowel syndrome.[4]
and 1 user experience i found on the net
I tried it while living in Egypt :
It comes in 50mg and the usual effect lasts 5 hours.It is usually taken in 100mg 3 times daily,and is not recomended to be taken befoe bedtime because it is the only "STIMULANT BENZODIAZEPINE" on the planet.
My experience is that it gives you a relaxed feeling combined with excellent concentration,motivation and sociability,without any muscle relaxant or any sedative,amnestic proporties + NO withdrawal effects at all
Its structure is fundementaly different from any other BZ (2,3 benzo) and,from my own experience I believe that it must be affecting dopamine in a way
The great thing about it is that you can take as needed for focus + anxiety or chronically without worrying about withdrawal.....
I know I might sound talking about a fantasy drug ,but the truth is that I only stopped it because I left Egypt and could not find it in the other countries I lived in......
Acta Pharm Hung. 1993 Mar;63(2):91-8.
Excerpts from the clinical-pharmacologic and clinical studies of Grandaxin
Szego J, Somogyi M, Papp E.
EGIS Gyogyszergyar Rt., Budapest.
The authors give a selection from the clinical-pharmacological and clinical studies of Grandaxin (tofizopam), an original Hungarian compound registered in 1976. Tofizopam, a 2,3-benzodiazepine derivative, differs from "classical" 1,4-benzodiazepines not only in chemical structure, but also in pharmacological and clinical-pharmacological properties. It is an anxiolytic without sedative-hypnotic, muscle relaxant and anticonvulsive effects. Tofizopam does not impair psychomotor and intellectual performance, like other benzodiazepines do, in the contrary, it has a mild stimulatory activity. It is potent in alleviating vegetative symptoms accompanying anxiety disorders. Tofizopam has a very low toxicity, mild side effects. The administration of tofizopam does not lead to physical or psychic dependence.
id be nice to try out, sounds interesting.
