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Extreme opioid tolerance - this is crazy

zorn

Bluelighter
Joined
Nov 11, 2001
Messages
5,636
Location
Kansas, USA
I was reading papers on ketamine/opioid analgesia last night and came across this paper which documents the most extreme case of opioid tolerance I've ever seen [1]. At its height this woman was receiving 7mg/hour of fentanyl (yes, milligrams) and was still pain.
This was a 22-year old woman in the last stages of terminal skin cancer; she had just rejected a white blood cell transfusion. Check it out:
"Five days after hospital admission her medication included hydromorphone 28 mg, fentanyl 350 µg, and lorazepam 6 mg per day."
"On ICU day 15, the patient was receiving 7000 µg/h of fentanyl and 10 mg/h of midazolam in addition to 100 mg methadone per day. Despite this regimen her pain control was inadequate and she complained of severe pain by nodding her head, grimacing, and fighting the ventilator."
"[On day 15] an initial attempt to convert fentanyl to an equipotent dose of hydromorphone (2065 mg) failed." (this was apparently done because she was receiving 3.4 liters/day of fentanyl infusion.)
"In an attempt to reduce opioid tolerance and improve analgesia, a ketamine infusion was started at 0.1 mg · kg-1 · hr-1 (8 mg/hr based on admission weight of 80 kg)... A taper of the fentanyl and midazolam infusions was initiated. Despite a lack of improvement of her overall medical condition, she progressively awoke over the next 5 days and on ketamine infusion day 6 (ICU day 21) she followed commands and indicated that she was comfortable by nodding her head appropriately to questions."
"The patient was transferred to the ward on ICU day 45 receiving only methadone at 300 mg/day"
Now this poor woman was intubated and ventilated, so respiratory depression wasn't an issue.. but the amount of opioids she was on is still truly amazing. Even more shocking is that 8mg/hr of ketamine made such a difference.
Comments anyone?
[1] Eilers H et al. (2001) The Reversal of Fentanyl-Induced Tolerance by Administration of "Small-Dose" Ketamine. Anaesthia and Analgesia 93:213-214.
 
my friends mom had severe back pain. Cuz she had an extra something or another which was eventually going to paralyse her. Anyway she was prescribed 100mg morphines, 5mg methadone, and little 500mg vials of ketamine.
 
Let's see, that would translate into 70 100ug/hour duragesic patches every three days, 700 patches a month...I wouldn't mind walking away with that perscription. You'd have a hell of a time getting it filled though!
"Yeah, uh, I need seventy boxes of duragesic, or you could just give me fourteen thousand Diluadid and a few crates of OxyContin - What? Why are the police here?" Of course the terminal cancer thing would kind of suck....Oh well, a small price to pay for the fine narcotics!
 
Oh well, a small price to pay for the fine narcotics!
/sarcasm on
Clearly, she thought it was worth the cancer too...
"Despite this regimen her pain control was inadequate and she complained of severe pain by nodding her head, grimacing, and fighting the ventilator."
/sarcasm off
 
Originally posted by MoFo_S:

Of course the terminal cancer thing would kind of suck....Oh well, a small price to pay for the fine narcotics!

Granted, large quantities of potent narcotics legitately perscribed would be nice, but when you are in extreme pain, I really doubt that you would enjoy them. Just wait until you have to watch someone close to you suffer through agonizing pain for months, and then get relief only through death. Then you may change your mind. But possible not. Not trying to flame, and I realize that mofo was trying to make a joke (hopefully), but after having watched family and friends suffer through cancer, those types of jokes piss me off. Terminal cancer is not something to joke about.
[ 06 February 2002: Message edited by: Grand Master of Somniferon ]
 
The secret encoded message in that was "Of course all of this is irrelevant because the horror of terminal cancer surely negates any joy that would otherwise be brought about by massive supplies of pharmaceutical narcotics, but this fact is so fucking obvious due to the extremeness of the situation that it does not need to be explicitly stated"
Maybe with my incredible talent for hidden sarcasm, I can go to the ER ODing on smack, and when they ask me what I took, I can just say "Uh, I'm a Narcan junkie who overdosed and is dying of horrible opioid antagonization" ... And they'll give me a big shot of oxymorphone and send me home!
 
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