Benzos Avizafone & Rilmazafone

[Dextro .45]

Brompton cocktail is a palliative elixir containing morphine, cocaine, ethanol, and other ingredients. So kind of but as a purist..

im stuck in bold btw

working class --- Be careful my guy; pack a large parachute for yourself.

Originally yes…however I have customized a Hybrid oral Brompton Cocktail due to chronic pain from RA

Even the original cocktail…..invented in the Royal Brompton Hospital in the United Kingdom in the 19th century

Morphine Sulphate can be replaced by Diacetylmorphine (Heroin), Hydromorphone (Dilaudid), Oxycodone or Methadone.

Cocaine can be replaced by Amphetamine, d-Amph, Ritalin (Methylphenidate) or d-Desoxyephedrine (Desoxyn/Methedrine) …even Phenmetrazine (Preludin), Biphetamine (Adderall), Benzphetamine

Chloroform water was used to raise volume for accurate dosing

Ethanol (usually Gin or Rum) & sweet juice to mask the bitter taste

Cannabis Indica

Now……MY own Brompton Cocktail

Methadone 100-125mg
Methylphenidate (Ritalin) 50-70mg IR
Diazepam (Valium) 30mg
Alprazolam (Xanax) 1mg
Pregabalin (Lyrica) 300mg
Ethanol (Gin) 2.oz drinks 4-6 over several hours

Fully tolerant male 6’ / 240 lbs ….taking for 10+ years …..Amazing for serious chronic pain

A POTENT Opioid Narcotic + a Dopaminergic Stimulant…..absolutely PARAMOUNT

 

[Working_Class]

what do you mean by fill out the gaps?? 0.25mg phenazolam dosed right when I wake up, to me feels like it drops off at maybe 8-10hrs past dosing, but i can tell its still active the next morning so ~24hrs past dosing. its half life is so long that i am skeptical about how long/sustainable daily dosing (just 1x/day) would be, but a low enough dose might plateau/stabilize out at a reasonable level.

it does pair well with both short and long-acting benzos, but unfortunately as you probably know, there aren't many options right now for short. ethylbrom reportedly feels a lot shorter and less sedating than brom, but who knows at this point- it may just be more subtle and last a long time too.

By fill up the gaps I mean one of those really long acting benzos is in you for something like 12 days, so frequent redosing would not really be the best way to go since it would jack up tolerance and just be an overall waste. It'd be good as like a once in awhile treat with a much shorter one to use in between those long-legged experiences. You know what I mean?


It's like if you just tried to use diazepam for every application. I don't think it would be that fantastic as landing gear. It synergizes really well with amphetamines say but it doesn't like "put me out" for example like alprazolam or Etizolam if I need it to just be over.


Unless I took some massive dose but then you'd be paying for it for like 3 days because then you be drowsy with the half-life being so incredibly long

 

[Working_Class]

Originally yes…however I have customized a Hybrid oral Brompton Cocktail due to chronic pain from RA

Even the original cocktail…..invented in the Royal Brompton Hospital in the United Kingdom in the 19th century

Morphine Sulphate can be replaced by Diacetylmorphine (Heroin), Hydromorphone (Dilaudid), Oxycodone or Methadone.

Cocaine can be replaced by Amphetamine, d-Amph, Ritalin (Methylphenidate) or d-Desoxyephedrine (Desoxyn/Methedrine) …even Phenmetrazine (Preludin), Biphetamine (Adderall), Benzphetamine

Chloroform water was used to raise volume for accurate dosing

Ethanol (usually Gin or Rum) & sweet juice to mask the bitter taste

Cannabis Indica

Now……MY own Brompton Cocktail

Methadone 100-125mg
Methylphenidate (Ritalin) 50-70mg IR
Diazepam (Valium) 30mg
Alprazolam (Xanax) 1mg
Pregabalin (Lyrica) 300mg
Ethanol (Gin) 2.oz drinks 4-6 over several hours

Fully tolerant male 6’ / 240 lbs ….taking for 10+ years …..Amazing for serious chronic pain

A POTENT Opioid Narcotic + a Dopaminergic Stimulant…..absolutely PARAMOUNT

I feel like that took some working up to, bravo

 

[Working_Class]

Etizolam Half Life Calculator - Graph and Multiple Doses

This etizolam half life calculator shows how etizolam accumulates and how long it stays in your body. Get dose and frequency with ease!

half-life-calculator.com

Sadly finished the batch. ~40 mg left. Nary enough for a good vibe but with a little beer, might be all good.

Now the search for new stash items begins...

I want a gram of this Ralmazafone, I need to see what the hell is up.witj Bromazolam, and Chlobromazolam sounds too good to not stock up on. A gram is like 4000 doses half life around 20+ hrs from reports (loose estimates).

Should be a legit lifetime supply

 

[pcplease]

bromazolam is gone. theres a new/novel form of substitution and true "RC" benzo, "ethylbromazolam" . vs how Brom and Phenazolam were developed decades ago. Yes it is extremely potent and with little/no tolerance 0.25mg is a moderate dose. 90-120min onset, but sublingual dosing helps a lot and some slowed breathing, laziness, starts in ~15min. but after that nothing for an hour and a half. lasts from morning to morning, feels "sober" after 8-12hr. meaning calm/no rebound anxiety whatsoever w/ that half life. which is nice compared to clonazolam, and lack of sedation vs bromazolam or especially flubromazolam.

 

[Working_Class]

bromazolam is gone. theres a new/novel form of substitution and true "RC" benzo, "ethylbromazolam" . vs how Brom and Phenazolam were developed decades ago. Yes it is extremely potent and with little/no tolerance 0.25mg is a moderate dose. 90-120min onset, but sublingual dosing helps a lot and some slowed breathing, laziness, starts in ~15min. but after that nothing for an hour and a half. lasts from morning to morning, feels "sober" after 8-12hr. meaning calm/no rebound anxiety whatsoever w/ that half life. which is nice compared to clonazolam, and lack of sedation vs bromazolam or especially flubromazolam.

There's tons of bromazolam around! But you're right, the Ethylbrom seems like the next in like doesn't it?

I've heard it's about half the potency and shorter acting.

I guess I'll have to see for myself soon

 

[pcplease]

by "gone" i just meant production has ceased china, and its availability towards the end of drying up in the US.

 

[Working_Class]

by "gone" i just meant production has ceased china, and its availability towards the end of drying up in the US.

Going, going, gone would be more like it haha. Stock up kids cause it's either gonna be impossible to find, subbed out or VERY expensive very soon.

Or gone as you say. Any of those

 

[pcplease]

Going, going, gone would be more like it haha. Stock up kids cause it's either gonna be impossible to find, subbed out or VERY expensive very soon.

Or gone as you say. Any of those

Powder in the US is gone outside of some extremely high markup, but w/ the US benzo market (read: xanax), means powder availability was rarely ever considerably cheaper than the same price to buy the chem already pressed into fake bars as anyone should expect to reasonably pay (under 3 figures) for a single gram of benzo powder when buying 1k minimum. So anyone wishing to stock up over here should forget about powder.

phenazolam bars have a foothold, though I'd hardly call it a replacement for brom/alp- They are for people who do not try to pass them off as alprazolam. Ethylbrom's reviews seem mixed but I am hopeful I will find a purpose for it if it is an effective, wakeful anxiolytic.

bromazolam and pyrazolam differ only in the phenyl vs pyridine ring. my fingers are crossed that ethylbromazolam is by pure Chinese chance, more like pyrazolam re: different BZD subreceptor affinities.

 

[notsmokeymcpot42088]

phenazolam is the next one I am looking at hard alright. That hasn't ceased production to anyone's knowledge? Why did bromazolam cease?

catch a ban or get scheduled in China or something? (I have enough trouble understanding the laws over here)

I feel the same way about 7 oh "Get it while it lasts; save it for when you are old and your doc dicks you over".

 

[pcplease]

phenazolam is the next one I am looking at hard alright. That hasn't ceased production to anyone's knowledge? Why did bromazolam cease?

catch a ban or get scheduled in China or something? (I have enough trouble understanding the laws over here)

I feel the same way about 7 oh "Get it while it lasts; save it for when you are old and your doc dicks you over".

it was banned last July in China, with a 6+mo notice of idk 100+ diff chems to be banned. bromazolam, flubromazepam i believe were the only new benzos.

phenazolam/"clobromazolam" was the immediate replacement, likely due to it already having been produced in China/known synthesis route, the name "clobromazolam" suggests to your average underinformed user that effects will be similar to bromazolam and/or flubromazolam. I was happy as I'd been in search for it for a couple years after first trying it. I stocked up quick, as cheap as it is per dose, knowing it was absolutely not a replacement for short-acting alprazolam or even the longer-acting, but similarly quick/hard-hitting bromazolam.

As such we have the novel ethylbromazolam, which is at minimum far weaker than phenazolam in effects, and moderately weaker by weight than bromazolam. It has yet to really take off as their are vendors who still have idk how many thousands/millions of bromazolam presses left in stock/to produce (again, the 2024 ban was announced MONTHS in advance, and as we saw with chinese alpraz, etiz, flualprazolam, clonazolam, people stock up if possible.

Phenazolam powder is still available via Chinese and domestic sources. Also fake bars, but this chem seriously deserves volumetric dosing as 0.25mg feels roughly as strong as 1-2mg clonazepam with a steep dose/response curve. Therapeutically very effective (as phenazepam was), but it can be very subtle at those to those without serious anxiety, BZD dependence, or other physical conditions which are affected by BZD's. Users might feel nothing from 0.25mg, "barely feel anything" from 0.5mg, and be stumbling/ blacked out for a full day from 1mg.

 

[notsmokeymcpot42088]

aye! Grazi so yes it is on super short supply too. Damn I will miss that one too I think. Shame China is banning them --- economically I would think it would be an opportunity but risk etc. Thank you for the info.

 

[Dextro .45]

Etizolam powder was sooo plentiful (REAL Etizolam is absolutely amazing)
Deschloroetizolam too

Diclazepam (2-Chloro Diazepam) - Delorazepam>>Lorazepam (Ativan)
Pro-Diazepam (Avizafone) prodrug to Valium (Diazepam)

Pregabalin & Gabapentin

 

[Dextro .45]

I have to agree %100 about Avizafone. I am ‘6.2 and 225lbs and very tolerant to benzodiazepines. And I MEAN tolerant. When I had a wisdom tooth removal done the dentist had to give me 5, 1/4mg Tiazolam tablets, I told him it might not be enough and after 20 min of waiting for the benz to start to take affect, the dentist was amazed how lucid and aware I was. He then had to give me another 2 1/4mg tabs before I was loopy enough to have my wisdom teeth removed. That being said, I weighed .04 on my scale or 40mg dissolved it into .75 mil of warm sterilized water and gave myself a SC jab into my belly chonk, and without a doubt 10 min or so later, (cannot be to sure on the time of onset) as I was very “lifted” as they say! Gotta admit it’s a great pro drug. And I also used to take the apotex brand 10mg of diazepam 5 tabs per day and they are SHIT! I never realized how impotent they really are! Would love to have some Kern brand if they are as potent as described. Just make sure you have a quality scale to measure your dose if you are benzodiazepine naïve. One that wieghs to the 100th of a gram or better yet 1000th. Either two or three 0’s after the decimal. Tanita scales are great just pricey.

Yeesssssss…….Canadian Apo-Tex brand Diazepam 10mg tablets are GARBAGE ……I can take 5 and be ….meh.

Spanish brand KERN Diazepam 10mg tiny non-scored light blue speckled tablets are REAL VALIUM …..2 to 3 tablets and I’m like jello & happy with no worries

Generic Apo-Tex 8.23mg per tablet
Kern Diazepam 11.9mg per tablet

Just guessing but generic is weak undercut shit….branded Pharma is pure on point, large players even synthesize their own API in house and have it analyzed for purity and weight, excipients used, pressed, etc

Some generics purchase their API’s over seas from China, India (no offence) cheapest price, not always 100% purity, often underweighted API in the tablets

Canadian generic Apo-Tex Diazepam 10mg are PURE TRASH lol

I will IM administer Avizafone (Pro-Diazepam) 60-80mg any day …..any day

 

[Dextro .45]

You are right as far as I can tell about avivazone. But as it doesn’t seem to provide a rush and diazepam has such high oral bioavailability, the expense—and it is expensive—doesn’t seem worth it.

$95 CDN ($80 USD roughly) for 1,000mg of Avizafone (Pro-Diazepam) ….so 10 doses of 100mg IM (High dose) realistically perhaps 15 doses of Avizafone for $100 CDN

Avizafone 22.5mg IM injection —— 0.5 to 0.7h C-max and Significantly higher levels in bloodstream
Diazepam 10mg oral —- 1h to 1.5 C-max and 1/3 peak serum levels in bloodstream as apposed to Avizafone

Significantly more water soluble, rapid acting pro-drug, IM injection into shoulder muscle onset in 10 - 15min with maximum serum levels in 30-45min ……rapidly penetrating the BBB with faster and higher Diazepam levels in all study participants with injection of Avizafone

42 Male / 6’ tall / 240lbs - tolerant individual…. 50 - 70mg of Avizafone (Pro-Diazepam) IM administered (which is roughly 30-50mg of Diazepam BUT with greater absorption, rapid onset, and significantly higher serum levels of Diazepam in CNS.

Oral Valium is also great, my #1 choice. Valium 10mg tablets & Xanax 2mg bars is all I’d require. 100,000 tablets each stored properly for long term storage…..or 100% pure pharmaceutical API powder of each substance

Ultimate supply of……every drug I’ll ever need and many taken daily for chronic pain

Methadone (40mg oral tablets & 100kg drums of API powder) Oxycodone/Diamorphine/Hydromorphone also)
Methylphenidate (Ritalin) - Desoxyn 5mg tablets
Diazepam (Valium) & Alprazolam (Xanax)
Pregabalin (Lyrica)
Clonidine 0.1mg tablets
Ketamine (crystal HCL & glass vials for injection)
LSD-25 (100ug tabs - many sheets)
MDMA - 100mg capsules if 100% pure pharmaceutical grade
Cannabis - Oils & flower (Indica - Sativa - Hybrid)
Depo-Testosterone 200mg IM (10ml glass vials - 1,000mg)
Ethanol - Gin & Rum + beer
Tobacco- Belmont premium cigarettes
Caffeine- Premium espresso & coffee

 

[notsmokeymcpot42088]

^ A man of simple tastes. Why not switch methadone out for H while we are dreaming and K for MXE -- That isn't a bad price for avazifone (Valhallium!) but bang for buck prolly better off with something in the Xanax potency range and if you behaved yourselve you may be able to afford that lifetime supply. The emergency ban on those 5 benzos just expired in the US too!! Huzzah!!

So no more need for the pro-drug loophole. (I am not a lawyer ftr) --- Are all of the lysergamines banned? You may be able to check that one off too. I don't see ethanol tobbacco caffeine or MJ going away. I know there was a Somethin methylphenidate analog but I can't vouch for it at all. Clonodine not sure if is scheduled but prolly not.

I say shoot for the stars! but avoid needles as much as possible haha

 

[canadianpeduser]

^ A man of simple tastes. Why not switch methadone out for H while we are dreaming and K for MXE -- That isn't a bad price for avazifone (Valhallium!) but bang for buck prolly better off with something in the Xanax potency range and if you behaved yourselve you may be able to afford that lifetime supply. The emergency ban on those 5 benzos just expired in the US too!! Huzzah!!

So no more need for the pro-drug loophole. (I am not a lawyer ftr) --- Are all of the lysergamines banned? You may be able to check that one off too. I don't see ethanol tobbacco caffeine or MJ going away. I know there was a Somethin methylphenidate analog but I can't vouch for it at all. Clonodine not sure if is scheduled but prolly not.

I say shoot for the stars! but avoid needles as much as possible haha

Does that mean there will be actual Valium back in the US

 

[Dextro .45]

The other one, prescribed in Japan….is weak grarbage from what I’ve read

Now, the other one…..on the other hand….one of the first “Blockbuster Drugs” Valium (Diazepam). Unfortunately not water soluble and IV/IM injections are painful and discomforting

France synthasized a water soluble pro-drug called Avizafone (Pro-Diazepam) which I have self administered 1,000mg bags X 4-6 over a few years ……simply Amazing compound. Amazing.

Even being marketed and sold to medical facilities were nurses and staff are physically & violently attacked and assaulted ….IM Midazolam is the current rapid acting benzodiazepine which is relatively fast onset & water soluble

But when minutes feel like hours , you need RAPID SEDATION.

Avizafone (Pro-Diazepam) 22.5mg IM injection = Diazepam 10mg oral tablet

My usual dose of Avizafone 50-70mg IM (roughly Valium 40mg) but with a 10-15min onset, with peak serum levels in 0.5 - 0.7h / v.s. 1.5h for oral Diazepam

Avizafone reaches a higher C-max and much faster
Oral administration sucks
SC injection is weak
IM injection is proper……designed ROA

 

[Dextro .45]

….and it’s the easiest shot you’ll ever give urself

Small glass vial (Dollar store arts & craft store) with aluminum screw cap top
Weight /and or place Avizafone powder in…..add clean bottled water (warm even slightly weak hot) for fast complete dissolving ….add with syringe 0.5ml water usually or 1ml max

Draw up clean water/Avizafone solution, no filter required, cleaned glass vial and pure clean water + API
Place needle gently near corner bottom and draw up solution

IM administered in shoulder muscle , in centre but slightly towards back 60/40
Proper needle gauge for IM injection 25Gauge diameter X 1” length needle (3ml but doesn’t matter, 1ml etc)


(My rig for depo-Testosterone 200mg is 22.5 Gauge and maybe 1.5” needle length …..for deep @$$ muscle IM shot lol, it’s a proper needle, bending the needle is tough…..not like some cheap 1ml 30gauge insulin syringe …..you can slam this bad boy rig into a grizzly bear neck with 1,000mg of Avizafone & 3,000mg Ketamine HCL and would do the job, not snapping, fat 3ml body ….add a G of Hydromorphone too lol …..that would be some needle packed with a punch … 1,000 lbs..Grizzly bear ok……human definitely fatal X 7 due to HM content

Such a rapid effective ROA. Eliminating first pass metabolism bypassing the liver, entering the bloodstream directly via IV injection of let’s say Diamorphine 100mg & Methedrine 20mg in a single syringe (my tolerance)

 

[Dextro .45]

How do you find deschloroetizolam? It is more easily available now than etiz. I find it a useful benzo, if not the very best.

You are 100% correct my friend

If you’re lucky enough to acquire near pharmaceutical grade, professionally synthesized Deschloroetizolam I’d acquire as much as financially possible

I had large gram quantities of both Etizolam and its Dechlorinated analog……to my surprise Deschloroetizolam was Significantly more pleasurable then Etizolam

Etizolam 1mg
Deschloroetizolam 6mg

It lasts longer also, same rapid onset of action 30-45min and 8-10h, as compared to Etizolams 6h or so. Deschloroetizolam gave me overwhelming robust anxiolytic & euphoric properties, as with Etizolam but more pronounced and noticeable……

In Canada I can still acquire Deschloroetizolam and Avizafone (Pro-Diazepam) but be aware, most Canadian vendors ONLY ship within Canada , as there is no customs to seize packages and cause heat for these Canadian Vendors . Canada Post, Xpresspost signature required + tracking number

Even my legally registered brand new Colt 1911 .45 ACP was handed to me by Canada Post…..the individual has ZERO idea what he was holding …….within Canada and you’re safe. No heat, no headaches

The batches of Deschloroetizolam 10-20 years ago (5,000mg +) I purchased I swear were as close to 98%+ near pharmaceutical grade compound. My 2mg micro scoop was used, 2 / 4 / 6mg dosing usually

Deschloroetizolam 6mg
Pregabalin 300mg
Dilaudid 2mg tablets X 6-8
Phenibut 1,000mg (3h onset) lasting 24 h with afterglow

Was a wonderful anxiolytic cocktail I enjoyed many times. Most all my compounded API substances were packed into empty large jel caps, 6-8 capsules in small plastic baggy

Later adding a dopaminergic stimulant including legally prescribe Ritalin (Methylphenidate) and illicit Cocaine, later on high quality Mephedrone - 4-MMC (950% increase in Serotonin & 500% increase in Dopamine)

Ritlain, Vyvanse, Dexedrine, Adderall XR are all Pharma stimulant meds I have been prescribed and used in therapeutic doses …..expect Ritalin 50-70mg IR with Ethanol (increasing d-threo-MPH by 40%) significantly enhancing euphoric pleasurable mood-boosting properties…..inhibiting over 50% of DAT dopamine transporters which is required to enduce euphoric effects in all test subjects

d-threo-Methylphenidate (Focalin) is the only isomer out of 4 possible isomers that inhibit DAT and induce release/increase in DAT/NET

Ritalin is 50/50 of both threo isomers ……..Ritalin 40mg = Focalin 20mg identical DAT inhibition

I hope you can acquire Deschloroetizolam my friend ………Avizafone (Pro-Diazepam) is my current go to, however I WISH I could acquire a very large quantity of pharmaceutical grade Diclazepam (2-Chloro Diazepam) which is like the Methadone of the benzodiazepine world, lasting longer than even Valium (Diazepam) itself