A paper about the SAR of novel 5-HT2A agonists

[Deleted member 170540]

This paper has been published this year, and contains information about a lot of exotic 5-HT2A ligands, like thieno analog of DMT and fluorinated tryptamines. Even a DMT analog with a carbon in place of indolic nitrogen is described as having affinity similar to the parent compound...

http://onlinelibrary.wiley.com/doi/10.1002/wmts.42/pdf

Just thought people would like to read this.

 

[Qadira]

Nice short review article. David Nichols has been a researcher in this field for many years. Thanks for posting.

 

[atrollappears]

Great read, thanks