Hi,
I am wondering what this data about Cyclizine means?
I am wondering what this data about Cyclizine means?
IC50: | SR-2B: IC50 = 0.37 nM (human); mAChR M5: IC50 = 0.63 nM (human); mAChR M1: IC50 = 0.68 nM (human); Histamine H1 Receptor: IC50 = 38 nM (human); SR-2A: IC50 = 225 nM (human) |
Ki Data: | Histamine H1 Receptor: Ki= 4.44 nM (human); SR-2A: Ki= 64 nM (human); mAChR M4: Ki= 119 nM (human); mAChR M3: Ki= 159 nM (human); Muscarinic acetylcholine receptor M1: Ki= 163 nM (human) Does it say that cyclizine is an antagonist at the receptors in this order? H1 > 5-HT2A > mAChR |