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  • Trip Reports Moderator: Xorkoth

(ETH-LAD/300µg) Experienced: Turned Inside-Out

perpetualdawn

Bluelighter
Joined
Nov 20, 2013
Messages
2,920
EXPERIENCE: 20+ years of psychedelics, including mushrooms, LSD, mescaline, 2C-x, LSZ, AL-LAD, one previous trial of ETH-LAD at a lower dosage of 150µg. Also have used various other psychedelics, dissociatives and other drugs.

TOLERANCE: No psychedelics used for ~7 weeks, so basically no tolerance.

SETTING: Mostly in my home, solo.

TIMELINE
(h0:00 = 8pm)
h0:00 300µg ETH-LAD sub buccal
h0:20 first alerts
h0:30 undeniably tripping
h2:00(ish) enter into a complete dissolution state, mind turned inside out
h6:00 back to earth, back to ?€œnormal?€ tripping level
h9:00 begin writing this report, still feeling diminishing effects.
h11:00 down to sleep, basically sober but tired.

INTRO
I wasn't properly prepared spiritually nor physically for this dose, and I experienced an overwhelming and complete dissolution of reality. My previous dose 8 weeks prior of 150µg ETH-LAD had been incredible, very strong, but easily manageable. I thought I could handle taking it up to 300µg. I was wrong. 300µg ETH-LAD turned me completely inside out, both metaphorically and physically. In my 20+ years of psychedelic usage, I've never experienced anything as extreme as the psychedelic dissolution from this 300µg of ETH-LAD. My reason for writing this report is twofold: to help myself to understand it, and to warn others regarding the potency of ETH-LAD.


THE TRIP
I put 2 of the current standard printed ETH-LAD blotters (300µg total) between my upper lip and gums, and then went for a walk to watch the sun set. As with my previous trial at 150µg, these tabs had an unmistakable sour taste, the same as how LSD tastes to me, but much stronger than any tab I've had before.

Within 20 minutes I could feel the first indication that the drug was working. By 30 minutes there was no denying that the ride had begun. By about 45 minutes I made my way back home as I could tell this was going to be a heavy trip.

I put on some meditative music on quietly, took care of a few minor chores around the house, started turning out the lights, which were already way too bright. Some neighbours were drinking and talking loudly, and it was very entertaining to hear their joyous laughter and chatter. By now it was about 1.5h in and I noticed that my neighbours voices were impossible to understand because they were echoing so heavily due to auditory hallucination. It was wild to listen to. After another half hour, they all went home, leaving a silent vacuum. I noticed that I was feeling a bit funny, trembling and a sense of malaise in my digestive tract.

At around 2h in I realized that I was going to have my first ever psychedelic vomit. In 20+ years of tripping, I've never once thrown up during a trip, not even from eating raw cactus. I partly blame the vomit on bad preparation food-wise, my body chemistry was way off from an overly salty bowl of pho I had eaten earlier.. Purge was needed. I had to think through the protocol for throwing up.. where are you supposed to throw up? How does it work? I fished the tabs out of my gums and noticed that they still had a lingering sour taste, so I'm not sure I had even absorbed all of the drug. The purge proceeded beyond emptying my stomach, on to profound retching up of a metaphysical/physical goop from what felt like the deepest pit of my guts, until there was absolutely nothing left in me. I felt a good bit better, but I could tell there was still something to unleash. At this point I realized I was in for a purgative kind of a trip.

I then tried to cleanse myself with a bath, but was hopeless. I managed to disrobe and get into the bathtub, but couldn't make any sense of how to operate the thing. Ended up having a few moments splashing around in half an inch of lukewarm bathwater as it ran down the drain. I couldn't get it together enough to draw a bath. I think I managed to partially brush my teeth, and then ended up on my livingroom floor wrapped in a towel.

From here on it's hard for me to remember where I was physically. I moved around a bit, mostly operating as a puddle on the floor. I wasn't really interfacing with the physical plane for about 3-4h. My mind was turned completely inside-out. I couldn't make sense of anything. I couldn't understand my senses, they were just streams of unintelligible, undifferentiated, synaesthetic information. I remember the sensation that these sense-streams were infinitesimally fine intertwined filaments.

This was a kind of psychedelic dissolution that I've imagined, and heard about, but in all my years of tripping had never experienced. It was overwhelming, uncomfortable, and confusing. I was in ?€œsquare root of negative one?€ land, where my mind was basically broken and turned inside out.

I did still have a have a grasp on shreds of reality here and there, but at many points my only anchor left was a faith that ?€œTIME EXISTS?€. This was an anchor I returned to several times, something that helped me not freak out under the absurd state of non-sense that I found myself in. It was a reminder or faith that eventually the state would subside and become more manageable. I was far enough out that I had no sense for what the quality of normal thought or experience was like, but I had the vague sense that there was something more reasonable that I would return to as time passed. But this notion of time, seemed more like a distant theory that I trusted in, because it was not something I felt I was experiencing. It wasn't like I felt like I was in a time-less state, or a state that was existed in opposition to time, it was more like time was a completely foreign, distant concept. But I knew somewhere that it was a real concept that I could count on.

Having established some kind of sane foundation, I became more comfortable with this scrambled abstract state, and explored some of the mental terrain.

I became aware that there exists what I can describe as ?€œintellectual black holes?€, asymptotic thought coordinates that occupy space radically outside of the bounds of logic and sense. Analogous to black holes of physics, these intellectual black holes are mental configurations or modes of thought that are possible for the human mind to go into, but from which information does not escape. Because they defy rationality and normal modes of thought so profoundly, it's impossible to store this information in memory. So when someone enters a ?€œblack hole?€ mode of thought, they appear as blackouts in retrospect as no memory can be formed of them. However, there is some way to cast some information out, by peering in from the edge, teetering on this event horizon, or stepping in a bit, and throwing a trail of breadcrumbs out. Then I realized that this idea of intellectual black holes wasn't just an abstract idea, but that I was actually orbiting around the edges of some intellectual black holes, in this barely comprehensible state of inside-out chaos.

I think I dipped into some of these black holes, because I can barely remember what all this was like. Or it's like I can remember the bits where I ?€œcame up for air?€, and there are a few gems of profound thought that came back to me the next day

There were some moments where survival instincts kicked in, and I was able to gather myself enough to do some simple things like drink some water from the tap, or cover my shivering naked body with my soggy towel. There were also moments of self-awareness where I was like ?€œohhhh so *this* is how people have pyschotic breaks on psychedelics?€. At times I felt like I was on the verge of running down the street naked save for a single sock on my head, yelling nonsense, like a nincompoop.

Around 2-3h after the onset of this complete psychic dissolution, I started to form actual thoughts that were marginally sensible - sensible enough to carry them forward from one moment-frame of awareness to the next. It was a relief to feel like I could hang my thoughts back onto the hooks of time. I thought it would be nice to make some mental notes to bring something back to earth. I thought the easiest way to explain the state I had been in would be to take whatever thought you could think of, but then think that thought inside out, so that instead of thinking that thought, you think the other side of that thought. I still have some glimmers of how that works, but I have to admit it doesn't make much sense now. Even at the time I knew it wouldn't.

I had a lot of spontaneous word-hallucinations. Strange goofy words came into my mind, things like: NurzleSnurf, WayambleSquanch, NoozleSkwoonch. NurzleSquirmf. These words seemed simultaneously hilarious and slightly disturbing.

Anyways, at 6h (about 4h after the beginning of the dissolution) I very abruptly found that I had touched back down on earth, into normal tripping territory with my feet on the ground.

It was exhilarating to be back to ?€œnormal?€ (actually still full blown tripping, with long tracers and typical psychedelia, but I had my ?€œego?€ or whatever back), I felt a bit lucky to be back in control and that I hadn't freaked out. It was a very sudden and distinct transition. I think my mind crossed some kind of threshold where the drug effects had diminished to the point where my mind was able to work coherently again. It was a bit like waking up or something.

I found some water, some fruit and then a beer to mellow into. I gathered myself, and went for a walk to get some fresh air and stretch my legs. By 9h into the trip I was nearing some kind of baseline, and I decided I should start writing this report before it all faded away, and then by 11h I tucked in to bed and was able to sleep easily.

Looking back the next day, I feel like I came down from that mountain of psychedelic dissolution, mostly empty handed, besides a few nonsense phrases. I'm disappointed in myself for not trusting my instincts going into this. I knew when I was dosing that I wasn't in quite the right place in body and spirit. I think it's easy to get away with these things being imperfect when the dose is lower, but at that high a dose there is no margin for error. And even if I had been better prepared leading up to it, it still would have been a dosage to unhinge my mind, in a way that I'm not sure I see any real value in.

On the other hand, I'm kind of glad I found out what a psychedelic overdose is like. It's pretty weird to unfold your mind like that. Never done that before. During the dissolution there were times when I was staring at something like what people might call the logos of perception and experience, and the parameters and bounds of reality, possibility and impossibility. One thing that really profoundly sat with me was the idea that mathematics is the most precise and high resolution study of the nature of reality, this plane of existence that we find ourselves in. I felt that I was wandering in the realm of the underlying structures of perception and existence, akin in some strange way to experiencing mathematical objects in a kind of fully synaesthetic manner.

Now that a couple of days have passed, I feel better about this trip. The negative aspects seem less important and I'm finding it easier to appreciate the wild ride, and am almost glad I put myself through this. However I have to remind myself that at the time, this was not a pleasant experience. I think it might be possible for me to enter a trip like this better prepared, and with someone to turn to if things got difficult. It is a little bit tempting to return to this realm under better circumstances, but I'm not sure if I ever will. I'm not sure that there's any point in turning your mind inside out like that.


SUMMARY/CONCLUSION
I've gained a healthy respect for the potency of ETH-LAD, and psychedelics in general. In my body at least, ETH-LAD is much stronger per µg than LSD.

For anyone wanting to explore this chemical, you should treat 150µg as your upper limit, and you might even want to try a 75µg dose first. My previous 150µg dose felt perfect. Strong, and perfect. I would never recommend someone takes 300µg of ETH-LAD, it was just way too much, at least for me. I imagine only the most hard-headed out there would need that kind of a dose.

I'm a bit concerned that my trip report might glamorize this kind of a high dose, because from the outside it might look like it was a pretty amazing ride. It *was* amazing, but it was not really what I would call a good experience, and I would not want to repeat this trip.

I feel like I got spanked, and learned a lesson in dosing safety. I wish I'd had a sitter or companion to turn to for help. I'm glad I kept my shit together enough to not do anything stupid. I feel like had I been a slightly less stoic person, slightly less experienced or had taken a bit more of the drug, I might have spent the night straightjacketed in a padded cell.

edit 2023: some character encoding seems to have gotten fucked up, all the apostrophes turned into ?€™, so fixed that. Still think about this crazy trip from time to time. I actually have some details to add in in retrospect, hope to make the time to do so.

Tagged by Xorkoth

substancecode_ethlad

substancecode_lysergamides

explevel_experienced

exptype_positive

exptype_difficult

roacode_sublingual
 
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Great report... Psychedelic over dose, maybe not, but it does sound like familiar territory with higher dosing ... Read' n into it, sounds like you raised your frequencies, welcome to the 5d reality
 
Yeah, great report indeed. I can totally relate to your experience. I only took 80-85 ug this weekend, and there actually was a point when I thought "holy shit" this just keeps getting more and more intense, but it didn't really in the end, there was just a while were it felt like it. So I can totally imagine how a high dose would leave you truly smashed.

Potent shit :) I can't wait to try 150 ug, but I doubt I'll go much higher.
 
Great report star. I am beginning to think more and more that it's not a good idea to push the dosages with these new lysergamides. Out of curiosity, did you feel as if you were overheating at all?
 
Thanks for checking out my trip report guys, it's kind of nice to know that some people read that.

Jammin: No I never felt like I was overheating during that trip.
 
Thanks for sharing, and in such great detail. High does definitely doesn't sound worthwhile, but I'm glad to have a sense of what it would be like.
 
This was a wonderful report, thank you for sharing! I can relate to this very much from higher dose LSD experiences.

When you spoke of the intellectual black holes and event horizons, it made me think back to an experience I had where I would slip into these out-of-body states where I was circling around the huge ring that was all darkness in the center, and the most beautiful patterns and imagery were flying by in the other direction. Those were very abstract but not actual blackouts; I have also had trips where I did blackout at times, and it wasn't as symbolic as that, but the most ridiculous parts of the experience definitely were when going into or coming out of that total loss of reality.

I will say, aside from the full blackouts which I do try to avoid, I do actually like being at that level when I intend to be there; I definitely think it's possible to treat it positively and get a lot of a reward out of it. Sometimes those states take some getting used to... but the impossibility of everything at that point is one of my favorite things about tripping. You've really piqued my interest here in fact.... Of all the psychedelics I've tried, so far 4-HO-DET is the one I've found to be the most potent in taking me to this impossible plane, and completely ripping reality apart along the way.... There are plenty of things it has less than other psychedelics, but when it comes your "square root of negative one" madness, for me it's unbeaten. And I bring it up specifically because of this wonderful chemical relationship....

168zuva.jpg

(Coincidence? o_O)
I haven't had the opportunity to try ETH-LAD yet but I have been waiting patiently for others to reveal its true nature, and now I am more interested in ever. Thank you again for sharing, this was very thorough and informative. :)
 
This was a fantastic read. You somehow managed to convey the utter confusion that occurs at high psychedelic doses in a way that is understandable and very relatable.

I actually squeeled out loud in excitement when you reffered to your mind space as the square root of -1 land. Awesome.

Glad you came out of the other side OK. Take care.
 
4-HO-DET and ETH-LAD aren't structurally very similar. Sure, it may look like that when purely looking at the structures as paintings, but when you take into account the electron wave functions, conformers (bond rotations and angles, placements) and things like that, plus the fact that 4-OH-DET is obviously missing the amide moiety, it becomes apparent that they aren't that similar after all. I don't know the pharmacodynamic profiles of either off the top of my head, but even if they are similar, I'd say it's just a coincidence.

Psychedelics are always intriguing, thanks for the nice post.
 
I must respectfully disagree. I believe that there is substantial scientific and anecdotal evidence to show that there is a significant overlap in the pharmacology and subjective effects of tryptamines and lysergamides, and I don't see the need to assume that there should be a better reason than their obvious molecular similarities. I also do not believe a lack of LSD's amide moiety is a deal breaker, as I am aware of at least one molecular docking prediction study which tested LSD, LSA, and agroclavine (which is just LSA without the amide part) and predicted similar receptor binding for all of them, and agroclavine was also found to have LSD-like behavioral and cortical effects in an old animal test from the late '50s. In relation to the parts of their molecules that they do share, I have to say that I am looking at them in a 3D viewer right now and they still look nearly identical. Do you have any evidence to what else could possibly cause the considerable overlap in their effects and pharmacology if not this?
 
I thought Eth-LAD had some similarities to 4-HO/AcO-MET which also has an ethyl group although less comformed. The colors especially reminded me of -MET (greens especially stood out).
 
That is very cool to hear as well as I absolutely love 4-HO-MET. :) I actually notice a heavy influence of green on it too, that's interesting. I do find it to have some things uniquely in common with 4-HO-DET as well, so I've really wondered if any of these attributes might carry over to ETH-LAD; hopefully some day I'll know.... I was just really interested in this trip report especially because the way perpetualdawn describes just being in total impossibility land really hit the nail on the head with describing how I feel about 4-HO-DET every time, it is an experience of compromised logic and reality and I often come out of it barely able to describe it in sane ways. 4-HO-MET I feel is unsurprisingly a little bit more like mushrooms and is not quite as far out there for me, but it does occasionally pass into that place and things get a little wonky or impossibly intricate. It's almost like a strange delirium, I wouldn't call it not psychedelic really but just sort of quirky; this is probably too subjective to identify with but for me personally it's most obvious feature is that 3D skeletal imagery is common for me on both of them and not other psychedelics, and it always correlates with that mindset. Anyway, thanks for sharing as well, I am definitely more intrigued in this one now!
 
Thats a fascinating idea re: the ethyl group and 4-HO-DET. When I tried ETH-LAD at the lower dosage of 150µg, I found it had some qualities that reminded me of 2C-E. I wonder if there really is something about the ethyl groups tickling the serotonin synapses in a particular way, or if it's just suggestion or our tendency to try to find patterns where there aren't necessarily any. I think 2C-E's ethyl is less likely to sit in the receptor site in the same position that ETH-LAD or 4-HO-DET does, but I really don't know how these molecules dock on the receptors.

In any case, I have to admit a fondness for ethyl groups. I'm intrigued to try out 4-HO-DET now.
 
That is very interesting as well, and I personally think it's worth considering that these molecules are simple enough that exposed ethyl groups could definitely cause some pharmacological overlaps even if it doesn't necessarily take place through the 5-HT2A receptor itself. For some time I have actually been fascinated by trying to figure out what these similarities may be, and though of course I cannot say what is and isn't actually relevant to the ultimate subjective effects of the psychedelic, I have noticed that between tryptamines, lysergamides, and phenethylamines (and other non-psychedelic bases as well like aminotetralins) there actually seems to be a pretty significant correlation between the length of exposed alkyl chains and dopamine (particularly D2-like) receptor binding. Something that stands out to me especially with the aminotetralins, which I have the most data of this kind on by far, is that while a propyl group has more affinity for them than an ethyl group, the ethyl group did confer the most selectivity for D2 between them, perhaps a good jumping off point for the near psychosis these psychedelics can provide? Who knows, but I think that the aminotetralins are probably similar enough structurally to the tryptamines that this pharmacological relationship is probably relevant even if that's not what it implies, especially given the known data that, for example, DPT is far more active at D2-like receptors than DMT.

As for the phenethylamines, that relationship may be a little more abstract, but it is known that they bind to at least D2 and D3 as well, but whether or not they do so significantly is debatable. PDSP data found the affinity numbers to be in the thousands for most of those versus the dozens for most of them at 5-HT2A, but I think it's interesting to note that they used a test ligand that supposedly will not properly label D2High or D3High binding, according to the guy who published said binding for LSD, arylcyclohexylamines, memantine, and a few other things. It was extremely difficult to dig up a paper comparing all D2, D2High, D3, and D3High for a single drug, and I was able to find it only for a sole antagonist (I believe it was iodosulpride but it's been quite a while since I read it now), but while I must say of course that what applies to this one drug clearly may not apply to others, I was quite shocked by what I was able to do with it. By getting ratios for low vs high affinity binding, I found this it was something like 77x more potent at D2High and 18x more potent at D3High (don't quote me on those numbers, I just remember it was close to that), and when I went to the PDSP data on phenethylamines to divide their given D2 and D3 affinity by those numbers assuming that they could have at least similar binding distribution, for the entire list it turned what seemed to be totally arbitrary and huge affinity numbers into values nearly identical(!) to their 5-HT2A binding; in fact, for 2C-E it was less than twice as potent at 5-HT2A compared to either D2 or D3.

So, while these numbers do rely on quite a bit of supposition and theory, it definitely made me a lot more curious about what all could be going on here. That's why I'm also very happy to see you mention 2C-E as well, because I only have experience with 2C-B and 2C-I, so unfortunately I am not in much a position to start exploring these theories myself on the phenethylamine side. I find the ethyl group psychedelics to be highly intriguing as well, and now you have made me even more anxious to get to try more of them some day. :) And I very much look forward to hearing your thoughts on 4-HO-DET if you ever get to try it!
 
Excellent report. Although I understand your trip was very unpleasant, I can't help but wonder about this "inside out" state of consciousness. I guess I'll never really know what it's like, but I wish I could take a peek into that world, if only for a few moments.

I *LOVE* your paragraph on "intellectual black holes". This is exactly the problem with DMT breakthroughs. They're very difficult to remember due to how alien they are.

At times I felt like I was on the verge of running down the street naked save for a single sock on my head, yelling nonsense, like a nincompoop.

LOL!! I have felt this way too, once.
 
Great report, thanks for sharing. :)

I became aware that there exists what I can describe as “intellectual black holes”, asymptotic thought coordinates that occupy space radically outside of the bounds of logic and sense. Analogous to black holes of physics, these intellectual black holes are mental configurations or modes of thought that are possible for the human mind to go into, but from which information does not escape. Because they defy rationality and normal modes of thought so profoundly, it’s impossible to store this information in memory. So when someone enters a “black hole” mode of thought, they appear as blackouts in retrospect as no memory can be formed of them. However, there is some way to cast some information out, by peering in from the edge, teetering on this event horizon, or stepping in a bit, and throwing a trail of breadcrumbs out. Then I realized that this idea of intellectual black holes wasn’t just an abstract idea, but that I was actually orbiting around the edges of some intellectual black holes, in this barely comprehensible state of inside-out chaos.

I feel this is what happened to me on my +4 2C-E trip years ago... thanks for putting that into words. I remember leading up to it, and I remember reaching a void where not even subjectivity existed anymore, the oneness existing outside of subjective experience. For just a moment. Then... I came to 30 minutes later, the peak gone. I am certain I continued to experience something but it was so abstract and apart from human experience that I have no way to recall it.
 
Phantastic report! Great to hear you came out mentally unscathed...


Great report star. I am beginning to think more and more that it's not a good idea to push the dosages with these new lysergamides. Out of curiosity, did you feel as if you were overheating at all?

Why did you ask this about Eth lad? Im curious because I and a few others I know got this effect from AL-LAD on every occasion Ive tried it accept when allergy testing
 
Very interesting report. It reminds me on my LSD experiences in the milligram-scale. The only difference I can see is that I walk a step further than you (or maybe your report isn't complete). I think I'll give eth-lad a try. Thanks for sharing your experience! :)
 
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