Butorphanol tartrate (Stadol)
Classification: Narcotic agonist/antagonist
Action/Kinetics: Has both narcotic agonist and antagonist properties. Analgesic potency is said to be up to 7 times that of morphine and 30-40 times that of meperidine. Overdosage responds to naloxone. After IV use, CV effects include increased PA pressure, pulmonary wedge pressure, LV end-diastolic pressure, system arterial pressure, pulmonary vascular resistance, and increased cardiac work load. Onset, IM: 10-15 min; IV: rapid; nasal: within 15 min. Duration, IM, IV: 3-4 hr; nasal: 4-5 hr. Peak analgesia, IM, IV: 30-60 min; nasal: 1-2 hr. t1/2, IM: 2.1-8.8 hr; nasal: 2.9-9.2 hr. Metabolized in the liver and excreted by the kidney. The drug has about 1/40 the narcotic antagonist activity as naloxone. A metered-dose nasal spray is now available.
Xyla-ject (xylazine) (liquid form)
This is an anesthetic, but not a discociative like Ketamine. It is not fun. DO NOT use this drug. It is only used in veterinary medicine now, as it has been proven to been too neurotoxic for human use.
Luminal (Phenobarbital sodium injection USP)
A barbituate... I have nodesire to play with this stuff.
SG