Pharmacology of Dipipanone

[TheJuner]

If there’s any good information about Dipipanone, specifically how it interacts with the my opioid receptors/binding affinity as well as the supposed NMDA antagonist properties it possesses could I get it? This abuse of Diconal has been well documented however I haven’t seen much in the way of it’s pharmacology.

 

[AlsoTapered]

Acta Chemica Scandinavica vol. 35b pp.613—619 The Crystal and Molecular Structure of Dipipanone Hydrochloride Hydrate. DOI: 10.3891/acta.chem.scand.35b-0613 a a	Barlein, Frode ;Mostad, Arvid ;Parker, Vernon D. ;Krogsgaard-Larsen, Povl ;Örn, Ulrika	Danish Chemical Society	1981
	Journal of the Forensic Science Society vol. 18 iss. 3-4 pp.262—0 Dipipanone, my Lord DOI: 10.1016/s0015-7368(78)71235-1 a a	T.L.		1978 July
	Journal of Chromatography A vol. 351 iss. none pp.249—258 Determination of dipipanone by high-performance liquid chromatography DOI: 10.1016/s0021-9673(01)83494-4 a a	S. Cathapermal; B. Caddy		1986 January		English
	Journal of Chromatography B: Biomedical Sciences and Applications vol. 424 iss. none pp.152—157 Measurement of dipipanone using capillary gas chromatography DOI: 10.1016/s0378-4347(00)81087-7 a a	Susan Paterson		1988 January
	Canadian Anaesthetists Society journal / Journal de la Société canadienne des anesthésistes vol. 6 iss. 1 pp.62—64 Report on the use of dipipanone hydrochloride as a postoperative analgesic DOI: 10.1007/bf03014196 a a	S. M. Campbell		1959 Janvier		French;English
	Journal of the Forensic Science Society vol. 5 iss. 4 pp.188—191 Acute Intoxication by Dipipanone DOI: 10.1016/s0015-7368(65)70264-8 a a	J.J. Taylor		1965 October
	Drug and Alcohol Review vol. 16 iss. 3 pp.221—226 Prescription of diamorphine, dipipanone and cocaine in England and Wales DOI: 10.1080/09595239800187401 a a	Dr LOUISE SELL; MICHAEL FARRELL; PHILIP ROBSON		1997 September 01		English
	British Journal of Clinical Pharmacology vol. 24 iss. 1 pp.43—50 Effects of triprolidine and dipipanone in the cold induced pain test, and the central nervous system of healthy volunteers. DOI: 10.1111/j.1365-2125.1987.tb03134.x a a	A Telekes; RL Holland; DA Withington; AW Peck		1987 July		English
	British Journal of Clinical Pharmacology vol. 24 iss. 6 pp.823—826 Dipipanone and nifedipine in cold induced pain; analgesia not due to skin warming. DOI: 10.1111/j.1365-2125.1987.tb03253.x a a	RL Holland; NE Harkin; SR Coleshaw; DA Jones; AW Peck; A Telekes		1987 December		English
	British Journal of Clinical Pharmacology vol. 33 iss. 4 pp.449—450 Pharmacokinetics of dipipanone after a single oral dose. DOI: 10.1111/j.1365-2125.1992.tb04066.x a a	S Paterson		1992 April		English
	British Journal of Pharmacology and Chemotherapy vol. 12 iss. 1 pp.97—99 ANALGESIC ACTIVITY OF DIPIPANONE HYDROCHLORIDE IN STUDENT VOLUNTEERS DOI: 10.1111/j.1476-5381.1957.tb01368.x a a	CAHAL, D. A.		1957 March
	The Lancet vol. 312 iss. 8087 pp.480 PSYCHOTIC SYMPTOMS AFTER DIPIPANONE DOI: 10.1016/S0140-6736(78)91493-9 a a	Bound, Denise; Greer, Steven		1978 August		English
	The Analyst (Royal Society of Chemistry) vol. 113 iss. 3 pp.385 Capillary gas chromatographic determination of cyclizine and dipipanone in biological fluids DOI: 10.1039/an9881300385 a a	Cathapermal, Segdabarum; Caddy, Brian		1988		English
	Palliative Medicine vol. 8 iss. 1 pp.63—65 Experience with dipipanone elixir in the management of cancer related pain - case study DOI: 10.1177/026921639400800111 a a	Faull, C.; McKechnie, E.; Riley, J.		1994 January		English
	Anesthesiology vol. 20 iss. 6 pp.902 DIPIPANONE DOI: 10.1097/00000542-195911000-00064 a a	Lamoureaux, L.		1959 November		English
	Anesthesiology vol. 20 iss. 2 pp.245 DIPIPANONE DOI: 10.1097/00000542-195903000-00127 a a	&NA;,		1959 March		English
	Anesthesiology vol. 18 iss. 4 pp.667 DIPIPANONE DOI: 10.1097/00000542-195707000-00080 a a	&NA;,		1957 July		English
	Survey of Anesthesiology vol. 3 iss. 5 pp.567???568 DIPIPANONE HYDROCHLORIDE (PIPADONE) AS A PRE-DELIVERY SEDATIVE AND ANALGESIC DOI: 10.1097/00132586-195910000-00030 a a	JOHNSTON, C. M.		1959 October
	Anesthesiology vol. 18 iss. 5 pp.801 DIPIPANONE DOI: 10.1097/00000542-195709000-00045 a a	&NA;, &NA;		1957 September		English
	Survey of Anesthesiology vol. 4 iss. 5 pp.458 PRELIMINARY CLINICAL STUDY OF DIPIPANONE HYDROCHLORIDE (PIPADONE) IN ANAESTHESIA DOI: 10.1097/00132586-196010010-00021 a a	LAMOUREUX, L.; SCHOONER, F.; TREMBLAY, L.		1960 October
	BMJ: British Medical Journal vol. 1 iss. 5027 pp.1092—1095 Dipipanone Hydrochloride as an Adjunct to Anaesthesia in Obstetrics and Surgery DOI: 10.1136/bmj.1.5027.1092 a a	Coleman, D. J. ;Levin, J. ;Jones, P. O.		1957 May 11		English
	Chemischer Informationsdienst vol. 13 iss. 12 ChemInform Abstract: THE CRYSTAL AND MOLECULAR STRUCTURE OF DIPIPANONE HYDROCHLORIDE HYDRATE DOI: 10.1002/chin.198212076 a a	BARLEIN, F.; MOSTAD, A.		1982 March 23
	BMJ: British Medical Journal vol. 2 iss. 6049 pp.1448—1448 Addictive abuse of dipipanone. DOI: 10.1136/bmj.2.6049.1448-a a a	James, I P ;Morgan, H G ;Gay, M		1976 December 11		English

All hotlinks.

I don't think it possesses any more NMDA activity than methadone, it's simply the fact that the infamous formulation was dipipanone + cyclizine. I'm old enough to have seen people put 3 tablets (pinks) in a 5mL barrel, add boiling water to dissolve it all and shoot it. No filtration. The effects are bizarre. You really do not want to be in ANY scene where people use Diconal. A guy I had known well for years accused me of stealing tablets he had injected 2 minutes before and if it hadn't been for the 1 other straight person in the room, it might well have kicked off.

All you need to know is that all of that crowd are dead with most not having even made it past 40.